Analysis of structure-activity relationships with the N-(3-acyloxy-2-benzylpropyl)-N'-[4-(methylsulfonylamino)benzyl]thiourea template for vanilloid receptor 1 antagonismLEE, Jeewoo; SU YEON KIM; LUNDBERG, Daniel J et al.Bioorganic & medicinal chemistry. 2004, Vol 12, Num 13, pp 3411-3420, issn 0968-0896, 10 p.Article

Antineoplastic agents 491,¹ Synthetic conversion of aaptamine to isoaaptamine, 9-demethylaaptamine, and 4-methylaaptaminePETTIT, George R; HOFFMANN, Holger; PETTIT, Robin K et al.Journal of organic chemistry. 2004, Vol 69, Num 7, pp 2251-2256, issn 0022-3263, 6 p.Article

Conformationally constrained analogues of diacylglycerol (DAG). Effect on protein kinase C (PK-C) binding by the isosteric replacement of Sn-1 and Sn-2 esters in DAG-lactonesKANG, Ji-Hye; CHUNG, Hye-Eun; SU YEON KIM et al.Bioorganic & medicinal chemistry. 2003, Vol 11, Num 12, pp 2529-2539, issn 0968-0896, 11 p.Article

N-(3-acyloxy-2-benzylpropyl)-N'-[4-(methylsulfonylamino)benzyl]thiourea analogues: Novel potent and high affinity antagonists and partial antagonists of the vanilloid receptorLEE, Jeewoo; LEE, Jiyoun; OH, Uhtaek et al.Journal of medicinal chemistry (Print). 2003, Vol 46, Num 14, pp 3116-3126, issn 0022-2623, 11 p.Article

N-4-t-Butylbenzyl 2-(4-methylsulfonylaminophenyl) propanamide TRPV1 antagonists: Structure-activity relationships in the A-regionKIM, Yong Soo; KIL, Min-Jung; JIN HEE LEE et al.Bioorganic & medicinal chemistry. 2012, Vol 20, Num 1, pp 215-224, issn 0968-0896, 10 p.Article

Analysis of structure-activity relationships for the 'b-region' of N-(3-acyloxy-2-benzylpropyl)-N'-[4-(methylsulfonylamino)-benzyl]thiourea analogues as vanilloid receptor antagonists: discovery of an N-hydroxythiourea analogue with potent analgesic activityLEE, Jeewoo; KANG, Sang-Uk; HA, Hee-Jin et al.Bioorganic & medicinal chemistry letters (Print). 2004, Vol 14, Num 9, pp 2291-2297, issn 0960-894X, 7 p.Article

N-[4-(methylsulfonylamino)benzyl]thiourea analogues as vanilloid receptor antagonists : Analysis of structure-activity relationships for the 'C-region'JEEWOO LEE; KANG, Sang-Uk; BLUMBERG, Peter M et al.Bioorganic & medicinal chemistry. 2004, Vol 12, Num 2, pp 371-385, issn 0968-0896, 15 p.Article

Structure―activity relationships and molecular modeling of the N-(3-pivaloyloxy-2-benzylpropyl)-N'-[4-(methylsulfonylamino)benzyl] thiourea template for TRPV1 antagonismBHONDWE, Rahul S; DONG WOOK KANG; BLUMBERG, Peter M et al.Bioorganic & medicinal chemistry letters (Print). 2012, Vol 22, Num 11, pp 3656-3660, issn 0960-894X, 5 p.Article

Analysis of structure-activity relationships for the 'B-region' of N-(4-t-butylbenzyl)-N'-[4-(methylsulfonylamino)benzyl ]- thiourea analogues as TRPV1 antagonistsLEE, Jeewoo; JIN, Mi-Kyoung; KIM, Sung-Eun et al.Bioorganic & medicinal chemistry letters (Print). 2005, Vol 15, Num 18, pp 4143-4150, issn 0960-894X, 8 p.Article

Structure-activity relationships of simplified resiniferatoxin analogues with potent VR1 agonism elucidates an active conformation of RTX for VR1 bindingLEE, Jeewoo; SU YEON KIM; WELTER, Jacqueline D et al.Bioorganic & medicinal chemistry. 2004, Vol 12, Num 5, pp 1055-1069, issn 0968-0896, 15 p.Article

Conformationally constrained analogues of N'-(4-tert-butylbenzyl)-N-(4-methylsulfonylaminobenzyl)thiourea as TRPV1 antagonistsLIM, Ju-Ok; JIN, Mi-Kyoung; RYU, Hyungchul et al.European journal of medicinal chemistry. 2009, Vol 44, Num 1, pp 322-331, issn 0223-5234, 10 p.Article

Non-vanillyl resiniferatoxin analogues as potent and metabolically stable transient receptor potential vanilloid 1 agonistsCHOI, Hyun-Kyung; CHOI, Sun; TRAN, Richard et al.Bioorganic & medicinal chemistry. 2009, Vol 17, Num 2, pp 690-698, issn 0968-0896, 9 p.Article

Stereospecific High-affinity TRPV1 Antagonists : Chiral N-(2-Benzyl-3-pivaloyloxypropyl) 2-[4-(methylsulfonylamino)phenyl]propionamide AnaloguesRYU, Hyungchul; JIN, Mi-Kyoung; TRAN, Richard et al.Journal of medicinal chemistry (Print). 2008, Vol 51, Num 1, pp 57-67, issn 0022-2623, 11 p.Article

Branched diacylglycerol-lactones as potent protein kinase C ligands and α-secretase activatorsLEE, Jeewoo; KANG, Ji-Hye; YOUNG HO KIM et al.Journal of medicinal chemistry (Print). 2006, Vol 49, Num 6, pp 2028-2036, issn 0022-2623, 9 p.Article

Macrocyclic diacylglycerol-bis-lactones as conformationally constrained analogues of diacylglycerol-lactones. Interactions with protein kinase CKANG, Ji-Hye; SU YEON KIM; JEEWOO LEE et al.Journal of medicinal chemistry (Print). 2004, Vol 47, Num 16, pp 4000-4007, issn 0022-2623, 8 p.Article

New bivalent PKC ligands linked by a carbon spacer: Enhancement in binding affinitySRIDHAR, Jayalakshmi; WEI, Zhi-Liang; NOWAK, Ireneusz et al.Journal of medicinal chemistry (Print). 2003, Vol 46, Num 19, pp 4196-4204, issn 0022-2623, 9 p.Article

2-(4-Methylsulfonylaminophenyl) propanamide TRPV1 antagonists: Structure―activity relationships in the B and C-regionsWEI SUN; KELIANG LIU; PEARCE, Larry V et al.Bioorganic & medicinal chemistry. 2012, Vol 20, Num 3, pp 1310-1318, issn 0968-0896, 9 p.Article

The SAR analysis of TRPV1 agonists with the α-methylated B-regionCHO, Yongsung; MYEONG SEOP KIM; HO SHIN KIM et al.Bioorganic & medicinal chemistry letters (Print). 2012, Vol 22, Num 16, pp 5227-5231, issn 0960-894X, 5 p.Article

Receptor activity and conformational analysis of 5'-halogenated resiniferatoxin analogs as TRPV1 ligandsKWANG SU LIM; DONG WOOK KANG; YONG SOO KIM et al.Bioorganic & medicinal chemistry letters (Print). 2011, Vol 21, Num 1, pp 299-302, issn 0960-894X, 4 p.Article

Halogenation of 4-hydroxy/amino-3-methoxyphenyl acetamide TRPV1 agonists showed enhanced antagonism to capsaicinDONG WOOK KANG; YONG SOO KIM; KWANG SU LIM et al.Bioorganic & medicinal chemistry. 2010, Vol 18, Num 22, pp 8092-8105, issn 0968-0896, 14 p.Article

α-Substituted N-(4 -tert-butylbenzyl ) -N'-[4 -(methylsulfonylamino )-benzyl]thiourea analogues as potent and stereospecific TRPV1 antagonistsCHUNG, Jae-Uk; SU YEON KIM; CHOI, Sun et al.Bioorganic & medicinal chemistry. 2007, Vol 15, Num 18, pp 6043-6053, issn 0968-0896, 11 p.Article

Analysis of structure-activity relationships for the 'A-region' of N-(4-t-butylbenzyl)-N'-[4-(methylsulfonylamino)benzyl]thiourea analogues as TRPV1 antagonistsLEE, Jeewoo; KANG, Sang-Uk; MIN, Kyung-Hoon et al.Bioorganic & medicinal chemistry letters (Print). 2005, Vol 15, Num 18, pp 4136-4142, issn 0960-894X, 7 p.Article

Antineoplastic agents. 499. Synthesis of hystatin 2 and related 1H-benzo[de][1,6]-naphthyridinium salts from aaptaminePETTIT, George R; HOFFMANN, Holger; HERALD, Delbert L et al.Journal of medicinal chemistry (Print). 2004, Vol 47, Num 7, pp 1775-1782, issn 0022-2623, 8 p.Article